平安! 发表于 2011-11-9 19:57 4 `, @. J. [- N7 Q/ `9 @
Pazopanib (100 mg/kg/day free base equivalent)
' j* i! D1 ~5 J- e6 k( i 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。/ F1 J6 a( U& u% w( Q+ I8 q; ^
搜索了一下,原料一大堆。+ U: w$ O3 {- B
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对不起!100mg/kg是用于移植瘤的,我弄错了。% m- g' k# U& z$ s
9 M$ \; m. k" \% D$ O以下是正版说明书的推荐用量。
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! A* [3 _8 ~& s, J8 d# @5 m$ ?--------------------- DOSAGE AND ADMINISTRATION ----------------# B' |! Z* ^9 f, [4 C. h% y) B
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
$ d1 Z% N. R3 S6 K3 L4 Y! r8 [* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
. I+ F: b9 L. u5 T' U1 h---------------------DOSAGE FORMS AND STRENGTHS --------------/ a* W4 W% y6 Y% M U: ~
200 mg tablets. (3) 1 u1 _# \1 [% c4 m" Q/ Z- k" w
-------------------------------CONTRAINDICATIONS------------------------ |