平安! 发表于 2011-11-9 19:57
& H- h. A4 E3 u$ n6 w( O! NPazopanib (100 mg/kg/day free base equivalent) ; k. a" _4 N: }
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
, X7 \& e! B+ ^ D搜索了一下,原料一大堆。
$ y" Q4 t+ G: K
! h" D8 b4 r6 r1 \1 V对不起!100mg/kg是用于移植瘤的,我弄错了。
( I5 d" m/ Q0 M! s* J, ?. P2 z$ j9 u8 L4 O# B( h; p8 u
以下是正版说明书的推荐用量。/ Q2 t6 J Y: T0 `# E1 R
, U# U/ n# B- u" q) a7 {# a0 U--------------------- DOSAGE AND ADMINISTRATION ----------------0 n7 |! [7 E4 ?6 W1 y( d0 l
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
6 N$ t7 U" T, n9 t. w( Y1 }* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) P/ H. I$ C' F5 M9 J/ M* p
---------------------DOSAGE FORMS AND STRENGTHS --------------+ k& M" S# V! h, L8 G
200 mg tablets. (3) 2 ]$ }- X8 _% e6 A
-------------------------------CONTRAINDICATIONS------------------------ |