平安! 发表于 2011-11-9 19:57 ( }5 d7 j% b7 C0 Z1 r# c
Pazopanib (100 mg/kg/day free base equivalent) - E3 a5 r2 N g* G
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。 s v, d; I9 e: \, p' w7 | ?
搜索了一下,原料一大堆。
2 R5 V+ |' e3 k/ A" F) b& [+ t, V h. @) ?: t: d
对不起!100mg/kg是用于移植瘤的,我弄错了。1 `% e) i5 _3 T1 z5 R8 I- j5 D
1 }" x; m# G* a0 g M) _; h
以下是正版说明书的推荐用量。. i0 L# z0 ?) A0 i4 V' T
; e4 L- t+ R# H
--------------------- DOSAGE AND ADMINISTRATION ----------------- b, d- L! S \+ L
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
) f8 J; \4 o3 o* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
, B Q% Z. ~1 U4 \/ ^" j---------------------DOSAGE FORMS AND STRENGTHS --------------
! n& s( F' {7 z8 y200 mg tablets. (3) 4 ^, M* X! L3 L, M/ y+ F8 e: G0 |6 \
-------------------------------CONTRAINDICATIONS------------------------ |